TheraRadar

Pharma Intelligence, Simplified

Data updated: Mar 10, 2026

ENVARSUS XR

TACROLIMUS
Immunology Approved 2015-07-10
2
Indications
--
Phase 3 Trials
10
Years on Market

Details

Status
Prescription
First Approved
2015-07-10
Routes
ORAL
Dosage Forms
TABLET, EXTENDED RELEASE

Companies

Active Ingredient: TACROLIMUS

ENVARSUS XR Approval History

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What ENVARSUS XR Treats

1 indications

ENVARSUS XR is approved for 1 conditions since its original approval in 2015. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Organ Rejection
Source: FDA Label

ENVARSUS XR Boxed Warning

MALIGNANCIES AND SERIOUS INFECTIONS Increased risk for developing serious infections and malignancies with ENVARSUS XR or other immunosuppressants that may lead to hospitalization or death [see Warnings and Precautions (5.1 , 5.2 )]. WARNING: MALIGNANCIES AND SERIOUS INFECTIONS See full prescribing information for complete boxed warning. Increased risk for developing serious infections and malignancies with ENVARSUS XR or other immunosuppressants that may lead to hospitalization or death. ( 5.1 ...

ENVARSUS XR Target & Pathway

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Target

IL-4 (Interleukin-4) Cytokine

A cytokine that promotes Th2 immune responses and IgE production. IL-4 drives allergic inflammation in atopic dermatitis and asthma. Blocking IL-4 (often together with IL-13) reduces the type 2 inflammation underlying these conditions.

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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

ENVARSUS XR FDA Label Details

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Indications & Usage

FDA Label (PDF)

ENVARSUS XR is a calcineurin-inhibitor immunosuppressant indicated for: The prophylaxis of organ rejection in de novo kidney transplant patients in combination with other immunosuppressants The prophylaxis of organ rejection in kidney transplant patients converted from tacrolimus immediate-release formulations in combination with other immunosuppressants 1.1 Prophylaxis of Organ Rejection in De Novo Kidney Transplant Patients ENVARSUS XR is indicated for the prophylaxis of organ rejection in kidney transplant patients in combination with other immunosuppressants [see Clinical Studies ]. 1.2 Pr...

⚠️ BOXED WARNING

WARNING: MALIGNANCIES AND SERIOUS INFECTIONS Increased risk for developing serious infections and malignancies with ENVARSUS XR or other immunosuppressants that may lead to hospitalization or death [see Warnings and Precautions (5.1 , 5.2 )]. WARNING: MALIGNANCIES AND SERIOUS INFECTIONS See full pre...

ENVARSUS XR Patents & Exclusivity

Latest Patent: Aug 2028

Patents (135 active)

US8664239 Expires Aug 30, 2028
US8685998 Expires Aug 30, 2028
US11123331 Expires May 30, 2028
US11110081 Expires May 30, 2028
US12083103 Expires May 30, 2028
US10864199 Expires May 30, 2028
US10166190 Expires May 30, 2028
US11419823 Expires May 30, 2028
US9549918 Expires May 30, 2028
US12403095 Expires May 30, 2028
+ 125 more patents
Source: FDA Orange Book

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.