TheraRadar

Pharma Intelligence, Simplified

Data updated: Mar 10, 2026

IDHIFA

ENASIDENIB MESYLATE
Oncology Approved 2017-08-01
2
Indications
--
Phase 3 Trials
2
Priority Reviews
8
Years on Market

Details

Status
Prescription
First Approved
2017-08-01
Routes
ORAL
Dosage Forms
TABLET

Companies

Active Ingredient: ENASIDENIB MESYLATE

IDHIFA Approval History

Loading approval history...

What IDHIFA Treats

1 indications

IDHIFA is approved for 1 conditions since its original approval in 2017. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Acute Myeloid Leukemia
Source: FDA Label

IDHIFA Boxed Warning

DIFFERENTIATION SYNDROME Patients treated with IDHIFA have experienced symptoms of differentiation syndrome, which can be fatal if not treated. Symptoms may include fever, dyspnea, acute respiratory distress, pulmonary infiltrates, pleural or pericardial effusions, rapid weight gain or peripheral edema, lymphadenopathy, bone pain, and hepatic, renal, or multi-organ dysfunction. If differentiation syndrome is suspected, initiate corticosteroid therapy and hemodynamic monitoring until symptom reso...

IDHIFA Competitors

Pro

1 other drug also targets IDH2. Compare mechanisms, indications, and trial activity.

Drug = Competitor name Company = Manufacturer N indic. = FDA-approved indications β†’ Date = Patent/exclusivity expiry

Competitors share the same molecular target (IDH2). Earlier expiry dates signal biosimilar/generic opportunities.

Drugs Similar to IDHIFA

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

DAURISMO
GLASDEGIB MALEATE
1 shared
Pfizer
Shared indications:
Acute Myeloid Leukemia
GRAFAPEX
TREOSULFAN
1 shared
MEDEXUS
Shared indications:
Acute Myeloid Leukemia
IDAMYCIN PFS
IDARUBICIN HYDROCHLORIDE
1 shared
Pfizer
Shared indications:
Acute Myeloid Leukemia
KOMZIFTI
ZIFTOMENIB
1 shared
KURA
Shared indications:
Acute Myeloid Leukemia
MYLOTARG
GEMTUZUMAB OZOGAMICIN
1 shared
Pfizer
Shared indications:
Acute Myeloid Leukemia
NEUPOGEN
FILGRASTIM
1 shared
Amgen
Shared indications:
Acute Myeloid Leukemia
NIVESTYM
FILGRASTIM-AAFI
1 shared
Pfizer
Shared indications:
Acute Myeloid Leukemia
NYPOZI
FILGRASTIM-TXID
1 shared
TANVEX BIOPHARMA USA INC
Shared indications:
Acute Myeloid Leukemia
ONUREG
AZACITIDINE
1 shared
Bristol-Myers Squibb
Shared indications:
Acute Myeloid Leukemia
RELEUKO
FILGRASTIM-AYOW
1 shared
KASHIV BIOSCIENCES LLC
Shared indications:
Acute Myeloid Leukemia
REVUFORJ
REVUMENIB CITRATE
1 shared
SYNDAX
Shared indications:
Acute Myeloid Leukemia
REZLIDHIA
OLUTASIDENIB
1 shared
RIGEL PHARMS
Shared indications:
Acute Myeloid Leukemia
RYDAPT
MIDOSTAURIN
1 shared
Novartis
Shared indications:
Acute Myeloid Leukemia
TIBSOVO
IVOSIDENIB
1 shared
SERVIER
Shared indications:
Acute Myeloid Leukemia
VANFLYTA
QUIZARTINIB DIHYDROCHLORIDE
1 shared
DAIICHI SANKYO INC
Shared indications:
Acute Myeloid Leukemia
VYXEOS
CYTARABINE
1 shared
JAZZ PHARMS THERAP
Shared indications:
Acute Myeloid Leukemia
XOSPATA
GILTERITINIB FUMARATE
1 shared
ASTELLAS
Shared indications:
Acute Myeloid Leukemia
ZARXIO
FILGRASTIM-SNDZ
1 shared
Novartis
Shared indications:
Acute Myeloid Leukemia
πŸ”¬

Active Pipeline

Pro

Ongoing clinical trials by development phase

Loading...
⭐

Key Completed Trials

Pro

Completed studies with published results, ranked by significance

Loading...
πŸ“Š

Trial Timeline

Full development history with FDA approval milestones

Loading...
Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

IDHIFA FDA Label Details

Pro

Indications & Usage

FDA Label (PDF)

IDHIFA is an isocitrate dehydrogenase-2 inhibitor indicated for the treatment of adult patients with relapsed or refractory acute myeloid leukemia (AML) with an isocitrate dehydrogenase-2 (IDH2) mutation as detected by an FDA-approved test . 1.1 Acute Myeloid Leukemia IDHIFA is indicated for the treatment of adult patients with relapsed or refractory acute myeloid leukemia (AML) with an isocitrate dehydrogenase-2 (IDH2) mutation as detected by an FDA-approved test.

⚠️ BOXED WARNING

WARNING: DIFFERENTIATION SYNDROME Patients treated with IDHIFA have experienced symptoms of differentiation syndrome, which can be fatal if not treated. Symptoms may include fever, dyspnea, acute respiratory distress, pulmonary infiltrates, pleural or pericardial effusions, rapid weight gain or peri...

IDHIFA Patents & Exclusivity

Latest Patent: Sep 2034

Patents (24 active)

US9732062 Expires Sep 16, 2034
US10093654 Expires Aug 1, 2034
US9738625 Expires Aug 1, 2034
US9512107 Expires Jan 7, 2033
US10294215 Expires Jan 7, 2033
US10610125 Expires Jun 21, 2030
+ 14 more patents
Source: FDA Orange Book

Want competitive intelligence?

See who's developing similar drugs and track their progress

View Pipeline Dashboard

Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.