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Data updated: Mar 10, 2026

VPRIV

VELAGLUCERASE ALFA
Rare Disease Approved 2010-02-26

VPRIV (velaglucerase alfa) is a hydrolytic lysosomal glucocerebroside-specific enzyme indicated for long-term enzyme replacement therapy in patients with type 1 Gaucher disease. This lysosomal storage disorder is characterized by the accumulation of glucocerebroside in the liver, spleen, and bone marrow, which can lead to organomegaly and hematologic complications. The therapy serves as a replacement for the deficient endogenous enzyme to manage the clinical features of the disease.

Source: FDA Label • Takeda • Hydrolytic Lysosomal Glucocerebroside-specific Enzyme

How VPRIV Works

Gaucher disease is caused by a deficiency in beta-glucocerebrosidase, an enzyme responsible for breaking down the sphingolipid glucocerebroside into glucose and ceramide. Without sufficient enzyme activity, glucocerebroside accumulates in the lysosomes of macrophages, forming "Gaucher cells" that infiltrate various organs. Velaglucerase alfa acts by catalyzing the hydrolysis of this accumulated glucocerebroside. This process reduces the volume of stored lipid, addressing the underlying cause of organ enlargement and blood-related symptoms.

Source: FDA Label
2
Indications
--
Phase 3 Trials
1
Priority Reviews
16
Years on Market

Details

Status
Prescription
First Approved
2010-02-26
Routes
INTRAVENOUS
Dosage Forms
INJECTABLE, POWDER

Companies

Active Ingredient: VELAGLUCERASE ALFA

VPRIV Approval History

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What VPRIV Treats

1 indications

VPRIV is approved for 1 conditions since its original approval in 2010. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Gaucher Disease
Source: FDA Label

VPRIV Boxed Warning

HYPERSENSITIVITY REACTIONS INCLUDING ANAPHYLAXIS Patients treated with enzyme replacement therapies have experienced life-threatening hypersensitivity reactions, including anaphylaxis. Anaphylaxis has occurred during the early course of enzyme replacement and after extended duration of therapy. Initiate VPRIV in a healthcare setting with appropriate medical monitoring and support measures, including access to cardiopulmonary resuscitation equipment. If a severe hypersensitivity reaction (e.g., a...

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Active Pipeline

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Ongoing clinical trials by development phase

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

VPRIV FDA Label Details

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Indications & Usage

FDA Label (PDF)

VPRIV is indicated for long-term enzyme replacement therapy (ERT) for patients with type 1 Gaucher disease. VPRIV is a hydrolytic lysosomal glucocerebroside-specific enzyme indicated for long-term enzyme replacement therapy (ERT) for patients with type 1 Gaucher disease.

⚠️ BOXED WARNING

WARNING: HYPERSENSITIVITY REACTIONS INCLUDING ANAPHYLAXIS Patients treated with enzyme replacement therapies have experienced life-threatening hypersensitivity reactions, including anaphylaxis. Anaphylaxis has occurred during the early course of enzyme replacement and after extended duration of ther...

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.